SCHEMBL7935113

SCHEMBL7935113

COc1cc([C@@H](O)CN)ccc1C

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 3/20 0.71
BLM P54132 3/20 0.69
PMP22 Q01453 1/20 0.69
CYP3A4 P08684 2/20 0.50
ADRA2A P08913 2/20 0.50
ADRA1A P35348 2/20 0.50
TSHR P16473 2/20 0.50
APEX1 P27695 3/20 0.49
TDP1 Q9NUW8 3/20 0.49
TAAR1 Q96RJ0 3/20 0.49
MAPT P10636 2/20 0.49
HPGD P15428 2/20 0.49
RECQL P46063 2/20 0.49
KDM4E B2RXH2 2/20 0.49
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
ADRB3 P13945 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1966507 0.86 NFKB1 (0.75) NFKB1BLMPMP22CYP3A4ADRA2A
SCHEMBL26092654 0.86 TSHR (0.53) NFKB1BLMPMP22CYP3A4TSHR
SCHEMBL29633151 0.86 NFKB1 (0.75) NFKB1BLMPMP22CYP3A4ADRA2A
SCHEMBL15921910 0.86 NFKB1 (0.75) NFKB1BLMPMP22CYP3A4ADRA2A
SCHEMBL7148550 0.86 NFKB1 (0.75) NFKB1BLMPMP22CYP3A4ADRA2A
SCHEMBL15965423 0.84 TSHR (0.70) NFKB1BLMPMP22CYP3A4TSHR
Hydrochloric Acid SCHEMBL8904803 0.84 BLM (0.76) NFKB1BLMPMP22CYP3A4ADRA2A
Normetanephrine SCHEMBL137755 0.83 NFKB1 (1.00) NFKB1BLMPMP22CYP3A4ADRA2A
Normetanephrine SCHEMBL4949341 0.83 NFKB1 (1.00) NFKB1BLMPMP22CYP3A4ADRA2A
Normetanephrine SCHEMBL29516838 0.83 NFKB1 (1.00) NFKB1BLMPMP22CYP3A4ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248573-B1 SULFONYLATING OR HALOGENATING A (S)-1-PHENYL-2-PROPANOL DERIVATIVE TO PRODUCE (S)-1-PHENYL-2-SUBSTITUTED PROPANE DERIVATIVE; CHEMICAL INTERMEDIATE FOR SYNTHESIS OF ANTIOBESITY DRUG DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-19 US disclosed
US-5902900-A OPTICAL PURITY, USE AS ANTI-OBESITY AGENTS DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-05-11 US disclosed
US-5679557-A Process of asymmetrically reducing 1-phenyl-2-oxo-propane derivatives with microorganisms DAICEL CHEMICAL INDUSTRIES, LIMITED (JP) 1997-10-21 US disclosed
EP-0627397-B1 Optically active 1-phenyl-2-substituted propane derivatives and methods of producing the same DAICEL CHEM (JP) 1997-01-02 EP disclosed
US-5508461-A ANTIOBESITY AGENTS DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-16 US disclosed
EP-0627397-A1 Optically active 1-phenyl-2-substituted propane derivatives and methods of producing the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-07 EP disclosed