SCHEMBL7935315

SCHEMBL7935315

Cc1ccc(-c2cc(C)ccc2/C=C/I)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.36
PSMB5 P28074 1/20 0.35
PELI1 Q96FA3 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MAOB P27338 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
HDAC7 Q8WUI4 1/20 0.33
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7935321 1.00 GRM2 (0.36) GRM2PSMB5PELI1NPC1RAB9A
SCHEMBL7935338 0.85 MAOB (0.34) GRM2PSMB5NPC1RAB9AMAOB
SCHEMBL7935342 0.85 MAOB (0.34) GRM2PSMB5NPC1RAB9AMAOB
SCHEMBL7931959 0.81 NFE2L2 (0.38) NPC1RAB9AMEN1KMT2AHDAC7
SCHEMBL7931961 0.81 NFE2L2 (0.38) NPC1RAB9AMEN1KMT2AHDAC7
SCHEMBL7929341 0.77 FYN (0.39) RAB9AMAOBKMT2AADORA3HDAC3
SCHEMBL7929345 0.77 FYN (0.39) RAB9AMAOBKMT2AADORA3HDAC3
SCHEMBL7930590 0.76 ALDH1A1 (0.43) GRM2PSMB5NPC1RAB9AMAOB
SCHEMBL15084634 0.71 PDE5A (0.36) KDM4EMAPTNFE2L2PTGS2NQO2
SCHEMBL13089999 0.71 PDE5A (0.39) KDM4EMAPTNFE2L2PTGS2NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0879814-B1 Triaromatic compounds, compositions containing them and uses thereof CT INTERNAT DE BR RECH S DERMA (FR) 2001-11-28 EP disclosed
US-6150413-A TREATMENT OF DERMATOLOGICAL, RHEUMATIC, RESPIRATORY, CARDIOVASCULAR, BONE AND OPHTHALMOLOGICAL DISORDERS, AS WELL AS MAMMALIAN SKIN AND HAIR CONDITIONS; 4-(4-(BIPHENYL-2-YL)BUT-3-EN-1-YNYL)BENZOIC ACID, FOR EXAMPLE CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (FR) 2000-11-21 US disclosed
EP-0879814-A1 Triaromatic compounds, compositions containing them and uses thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (C.I.R.D. GALDERMA) (FR) 1998-11-25 EP disclosed