SCHEMBL7937327

SCHEMBL7937327

NC(=O)c1ccc(C2C=CC=CC2)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.37
GLA P06280 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HIF1A Q16665 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GSK3B P49841 1/20 0.35
SIRT6 Q8N6T7 2/20 0.33
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
LCK P06239 1/20 0.33
APP P05067 1/20 0.32
AURKA O14965 1/20 0.31
PDPK1 O15530 1/20 0.31
RPS6KB1 P23443 1/20 0.31
ADORA3 P0DMS8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30615382 0.73
SCHEMBL22004261 0.73 CA12 (0.40) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL18296234 0.73 KMT2A (0.60) KMT2AKDM4EGLAHTTSMN1; SMN2
SCHEMBL23161981 0.70 MEN1 (0.33) KMT2A
SCHEMBL23447069 0.70 MEN1 (0.33) KMT2A
SCHEMBL12993026 0.70 MEN1 (0.33) KMT2A
SCHEMBL21586650 0.70 SLC6A2 (0.39) KDM4EHTTKDM1A
SCHEMBL13211931 0.68 TSHR (0.43) SMN1; SMN2TDP1TSHR
SCHEMBL3736028 0.68 KMT2A (0.54) KMT2AKDM4EGLAHTTSMN1; SMN2
SCHEMBL28235965 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025235-A1 SELECTIVE LIGANDS FOR THE DOPAMINE 3 (D3) RECEPTOR AND METHODS OF USING THE SAME REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2010-03-04 WO disclosed