SCHEMBL7938441

SCHEMBL7938441

COc1ccc(N)cc1C1CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 3/20 0.46
USP2 O75604 1/20 0.46
HTR2A P28223 2/20 0.45
MAPT P10636 3/20 0.44
CYP19A1 P11511 3/20 0.44
GAA P10253 2/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
HTR2C P28335 2/20 0.43
NR4A1 P22736 1/20 0.43
ADRA1A P35348 2/20 0.41
NR3C1 P04150 1/20 0.40
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11819421 0.91 HTR2A (0.53) KDM4EALDH1A1USP2HTR2AMAPT
SCHEMBL6815422 0.88 HTR2C (0.61) HTR2AHTR2C
SCHEMBL7029357 0.87 QDPR (0.52) KDM4EALDH1A1USP2HTR2AMAPT
SCHEMBL2570589 0.85 MAPT (0.48) KDM4EALDH1A1USP2HTR2AMAPT
SCHEMBL6924205 0.84 ABCB1 (0.43) KDM4EALDH1A1MAPTLMNAADRA1A
SCHEMBL6717514 0.83 EHMT2 (0.42) KDM4EALDH1A1HTR2AMAPTLMNA
SCHEMBL6714974 0.82 ABCB1 (0.47) KDM4EALDH1A1HTR2AMAPTLMNA
SCHEMBL8536319 0.81 SLC6A2 (0.44) KDM4EALDH1A1MAPTLMNANR4A1
SCHEMBL7880812 0.81 HTR2A (0.47) HTR2AHTR2C
SCHEMBL4771915 0.81 MEN1 (0.52) ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010051236-A1 ISONICOTINAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-05-06 WO disclosed