SCHEMBL7938906

SCHEMBL7938906

Nc1nc(N)c2ncnc(N)c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.45
LIMK1 P53667 5/20 0.39
CDK2 P24941 4/20 0.39
CDC7 O00311 4/20 0.39
CDK1 P06493 3/20 0.39
CDK5 Q00535 2/20 0.39
PLK4 O00444 2/20 0.39
AURKA O14965 2/20 0.39
ROCK2 O75116 2/20 0.39
PIM1 P11309 2/20 0.39
PRKACA P17612 2/20 0.39
RPS6KB1 P23443 2/20 0.39
MARK3 P27448 2/20 0.39
FLT4 P35916 2/20 0.39
KDR P35968 2/20 0.39
CSNK1D P48730 2/20 0.39
GSK3A P49840 2/20 0.39
STK3 Q13188 2/20 0.39
ROCK1 Q13464 2/20 0.39
DYRK1A Q13627 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7940046 0.79 ADORA2A (0.48) ADORA2ACDK2CDK1CCNB1CCNE1
SCHEMBL7930934 0.77 CDK1 (0.43) ADORA2ALIMK1CDK2CDC7CDK1
SCHEMBL7942505 0.77 LMNA (0.45) ADORA2AMAP4K4PI4KAPI4K2BPI4K2A
SCHEMBL16094493 0.69 HSP90B1 (0.33) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL5989622 0.69 ADORA2A (0.41) ADORA2ACDK2CDK1DYRK1ACSNK1A1
SCHEMBL6416647 0.68 EGFR (0.44) MAP4K4PI4KAPI4K2BPI4K2API4KB
SCHEMBL4815326 0.67 ADORA2A (0.41) ADORA2ACDK2CDK1CCNB1CCNE1
SCHEMBL5386086 0.67 ADORA2A (0.55) ADORA2AKDM4EALDH1A1MAPTHPGD
SCHEMBL22715826 0.66 ADORA2A (0.41) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL22715627 0.66 ADORA2A (0.37) ADORA2AMAP4K4PI4KAPI4K2BPI4K2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968329-A1 NOVEL BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF USING SAME Galleon Pharmaceuticals, Inc. (US) 2016-01-20 EP disclosed
WO-2014151462-A1 NOVEL BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF USING SAME GALLEON PHARMACEUTICALS, INC. (US) 2014-09-25 WO disclosed
US-6232312-B1 ADMINISTERING A COMBINATION OF INDENE AND PYRIMIDO(5,4-D)PYRIMIDINE DERIVATIVES TO TREAT PREPANCREATIC CANCER CELL PATHWAYS, INC. 2001-05-15 US disclosed