SCHEMBL7939608

SCHEMBL7939608

COc1cc(C(O)C(=O)NCc2ccc(O)c(O)c2)ccc1O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 3/20 0.57
ERCC4 Q92889 3/20 0.57
TSHR P16473 3/20 0.57
BLM P54132 3/20 0.57
NPSR1 Q6W5P4 2/20 0.57
CYP3A4 P08684 5/20 0.50
ALOX15 P16050 3/20 0.50
KDM4E B2RXH2 2/20 0.50
GAA P10253 2/20 0.50
RAB9A P51151 1/20 0.50
GLS O94925 1/20 0.50
CYP1A2 P05177 4/20 0.49
ALDH1A1 P00352 3/20 0.49
CYP2D6 P10635 3/20 0.49
CYP2C9 P11712 3/20 0.49
CYP2C19 P33261 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
TRPV1 Q8NER1 2/20 0.49
PMP22 Q01453 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7947186 0.95 BLM (0.53) ERCC1ERCC4TSHRBLMNPSR1
SCHEMBL7939628 0.90 TSHR (0.57) TSHRBLMNPSR1CYP3A4ALOX15
SCHEMBL7947240 0.88 TYR (0.57) TSHRBLMNPSR1ALOX15KDM4E
SCHEMBL7947252 0.87 ERCC1 (0.65) ERCC1ERCC4TRPV1
SCHEMBL8108684 0.82 ALOX15 (0.59) ERCC1ERCC4TSHRBLMNPSR1
SCHEMBL17667848 0.80 CYP3A4 (0.60) ERCC1ERCC4TSHRBLMNPSR1
SCHEMBL4947604 0.80 CYP3A4 (0.60) ERCC1ERCC4TSHRBLMNPSR1
SCHEMBL6364316 0.79 ERCC1 (0.72) ERCC1ERCC4TSHRCYP3A4ALOX15
SCHEMBL7939631 0.79 ERCC1 (0.54) ERCC1ERCC4TSHRBLMCYP3A4
SCHEMBL3872413 0.77 CYP1A2 (0.57) TSHRBLMNPSR1CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265611-B1 USE AS ANTIOXIDANTS OR FREE-RADICAL SCAVENGERS IN COSMETICS AND PHARMACEUTICALS AND FOODS HAARMANN & REIMER GMBH (DE) 2001-07-24 US claimed
EP-1029849-A1 Hydroxymandelamides of phenolic amines HAARMANN & REIMER GMBH (DE) 2000-08-23 EP claimed
US-6265611-B1 USE AS ANTIOXIDANTS OR FREE-RADICAL SCAVENGERS IN COSMETICS AND PHARMACEUTICALS AND FOODS HAARMANN & REIMER GMBH (DE) 2001-07-24 US disclosed
EP-1029849-A1 Hydroxymandelamides of phenolic amines HAARMANN & REIMER GMBH (DE) 2000-08-23 EP disclosed