SCHEMBL7939742

SCHEMBL7939742

N#Cc1ccc(C2N=C(N)c3ccccc3N2)cc1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 11/20 0.69
NOS1 P29475 1/20 0.45
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
LRRK2 Q5S007 1/20 0.39
CCKBR P32239 1/20 0.34
TSHR P16473 1/20 0.33
MAOB P27338 1/20 0.33
KDR P35968 1/20 0.32
MYB P10242 1/20 0.32
IDO1 P14902 1/20 0.32
CHEK1 O14757 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8381026 0.99 NOS2 (0.68) NOS2NOS1NPC1RAB9ALRRK2
SCHEMBL7802794 0.82 NOS2 (1.00) NOS2NOS1
Hydrochloric Acid SCHEMBL8378309 0.81 NOS2 (0.96) NOS2NOS1
SCHEMBL7802808 0.78 NOS2 (0.78) NOS2NOS1NPC1RAB9A
Hydrochloric Acid SCHEMBL8381045 0.77 NOS2 (0.76) NOS2NOS1NPC1RAB9A
SCHEMBL7940647 0.77 NOS2 (0.69) NOS2NOS1NPC1RAB9ALRRK2
SCHEMBL7806725 0.74 NOS2 (0.66) NOS2NOS1LRRK2
Hydrochloric Acid SCHEMBL8379923 0.73 NOS2 (0.64) NOS2NOS1LRRK2
SCHEMBL23939363 0.67 LRRK2 (0.43) NPC1RAB9ALRRK2CCKBRKDR
SCHEMBL7938376 0.67 NOS2 (0.59) NOS2NOS1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed
CN-1204327-A Pharmaceutically active quinazoline compounds ASTRA PHARMA PROD (GB) 1999-01-06 CN disclosed