SCHEMBL7940647

SCHEMBL7940647

CN(C)c1ccc(C2N=C(N)c3ccccc3N2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 10/20 0.69
ALDH1A1 P00352 5/20 0.48
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
MAPT P10636 3/20 0.48
KDM4E B2RXH2 2/20 0.48
TP53 P04637 2/20 0.48
HPGD P15428 2/20 0.48
GLA P06280 1/20 0.48
GAA P10253 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
RUNX1 Q01196 1/20 0.48
CBFB Q13951 1/20 0.48
HSD17B10 Q99714 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
NOS1 P29475 1/20 0.45
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8381067 0.99 NOS2 (0.68) NOS2ALDH1A1MEN1KMT2AMAPT
SCHEMBL7802794 0.82 NOS2 (1.00) NOS2ALDH1A1MEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL8378309 0.81 NOS2 (0.96) NOS2ALDH1A1MEN1KMT2AKDM4E
SCHEMBL7802808 0.78 NOS2 (0.78) NOS2ALDH1A1MAPTKDM4ETP53
Hydrochloric Acid SCHEMBL8381045 0.77 NOS2 (0.76) NOS2ALDH1A1MAPTKDM4ETP53
SCHEMBL7939742 0.77 NOS2 (0.69) NOS2NOS1NPC1RAB9ALRRK2
Hydrochloric Acid SCHEMBL8381026 0.75 NOS2 (0.68) NOS2NOS1NPC1RAB9ALRRK2
SCHEMBL7806725 0.74 NOS2 (0.66) NOS2ALDH1A1MEN1KMT2AMAPT
Hydrochloric Acid SCHEMBL8379923 0.73 NOS2 (0.64) NOS2ALDH1A1MEN1KMT2AMAPT
SCHEMBL7803338 0.69 NOS2 (1.00) NOS2KDM4EGAAHSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed
CN-1204327-A Pharmaceutically active quinazoline compounds ASTRA PHARMA PROD (GB) 1999-01-06 CN disclosed