SCHEMBL7940883

SCHEMBL7940883

CCOC(=O)N1CCC2(CC1)N=C(N)c1c(F)cccc1N2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 10/20 1.00
NOS1 P29475 8/20 1.00
NOS3 P29474 2/20 1.00
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.46
POLB P06746 1/20 0.42
ALOX15 P16050 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KCNH2 Q12809 1/20 0.42
BRD4 O60885 1/20 0.41
LMNA P02545 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
OPRD1 P41143 2/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8379951 0.99 NOS2 (0.98) NOS2NOS1NOS3ALDH1A1KDM4E
SCHEMBL7931849 0.93 NOS2 (0.87) NOS2NOS1NOS3ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL8379849 0.92 NOS2 (0.85) NOS2NOS1NOS3ALDH1A1KDM4E
SCHEMBL7931756 0.91 NOS2 (0.84) NOS2NOS1NOS3ALDH1A1KDM4E
SCHEMBL7938128 0.90 NOS2 (0.82) NOS2NOS1NOS3ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL8376625 0.90 NOS2 (0.82) NOS2NOS1NOS3ALDH1A1KDM4E
SCHEMBL7931779 0.90 NOS2 (0.82) NOS2NOS1NOS3ALDH1A1KDM4E
SCHEMBL7804468 0.90 NOS2 (0.82) NOS2NOS1NOS3ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL8380988 0.90 NOS2 (0.81) NOS2NOS1NOS3ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL8518505 0.90 NOS2 (0.81) NOS2NOS1NOS3ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed