SCHEMBL794177

SCHEMBL794177

COc1cc(S(=O)(=O)Nc2cccc(-c3nnn[nH]3)c2)ccc1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.50
CA9 Q16790 1/20 0.50
TP53 P04637 4/20 0.47
PLAU P00749 1/20 0.47
HTT P42858 4/20 0.47
LMNA P02545 3/20 0.47
ALDH1A1 P00352 2/20 0.47
TSHR P16473 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
PKM P14618 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALOX12 P18054 1/20 0.46
PFKFB4 Q16877 2/20 0.46
PFKFB3 Q16875 3/20 0.45
MAPT P10636 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
NTRK1 P04629 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL794304 0.83 PFKFB3 (0.63) HTTLMNAALDH1A1PFKFB4PFKFB3
SCHEMBL27943370 0.83 MMP2 (0.59) TP53HTTLMNAALDH1A1PKM
SCHEMBL793607 0.82 PFKFB4 (0.64) HTTLMNAALDH1A1PFKFB4PFKFB3
SCHEMBL793433 0.81 PFKFB4 (0.67) TP53PLAUHTTLMNAALDH1A1
SCHEMBL6792745 0.81 CA12 (0.74) CA12CA9PLAUHTTLMNA
SCHEMBL793299 0.80 PFKFB3 (0.65) PLAUHTTLMNATSHRPKM
SCHEMBL793359 0.80 PFKFB3 (0.68) TP53PLAUHTTLMNAALDH1A1
SCHEMBL793619 0.77 PFKFB3 (0.71) TP53LMNAPKMPFKFB4PFKFB3
SCHEMBL793788 0.77 PFKFB3 (0.59) TP53LMNAPKMPFKFB4PFKFB3
SCHEMBL795004 0.76 PFKFB3 (0.60) TP53LMNAPFKFB4PFKFB3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616450-A2 SULFONAMIDE COMPOUNDS Kancera AB (SE) 2013-07-24 EP disclosed
WO-2012035171-A2 NEW COMPOUNDS KANCERA AB (SE) 2012-03-22 WO disclosed