SCHEMBL7942015

SCHEMBL7942015

C#CCC(=O)Nc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.66
CYP1A2 P05177 1/20 0.66
CYP2D6 P10635 1/20 0.66
EPHX2 P34913 2/20 0.57
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
MAPT P10636 3/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
HTT P42858 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
TP53 P04637 1/20 0.52
EPHX1 P07099 1/20 0.52
TSHR P16473 1/20 0.52
CDK9 P50750 1/20 0.52
CLK4 Q9HAZ1 1/20 0.52
KDM1A O60341 1/20 0.52
GAA P10253 1/20 0.52
SCN1A P35498 1/20 0.52
SCN2A Q99250 1/20 0.52
SCN3A Q9NY46 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15612337 0.94 CYP1A2 (0.60) CYP3A4CYP1A2CYP2D6EPHX2MEN1
SCHEMBL15612046 0.89 CYP1A2 (0.55) CYP3A4CYP1A2CYP2D6EPHX2MEN1
SCHEMBL8375614 0.83 EPHX2 (0.57) CYP3A4CYP1A2CYP2D6EPHX2MEN1
SCHEMBL4813925 0.82 CYP3A4 (0.81) CYP3A4CYP1A2CYP2D6EPHX2MEN1
SCHEMBL10784058 0.82 EPHX2 (0.52) CYP3A4CYP1A2CYP2D6EPHX2MEN1
SCHEMBL11412618 0.82 EPHX2 (0.55) EPHX2MAPTL3MBTL1HTTSMN1; SMN2
SCHEMBL1260216 0.82 SMN1; SMN2 (0.62) CYP1A2EPHX2MEN1KMT2AMAPT
SCHEMBL11250189 0.80 SMN1; SMN2 (0.60) CYP3A4CYP1A2CYP2D6EPHX2MEN1
SCHEMBL22231489 0.80 GAA (0.59) MEN1KMT2AMAPTSMN1; SMN2TP53
SCHEMBL1689206 0.80 EPHX2 (0.68) CYP3A4EPHX2MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0834499-B1 Process for the preparation of aromatic vinyl compounds DAINIPPON INK & CHEMICALS (JP) 2001-07-25 EP disclosed
EP-0834499-A1 Process for the preparation of aromatic vinyl compounds DAINIPPON INK AND CHEMICALS, INC. (JP) 1998-04-08 EP disclosed
US-4661632-A Halogenopropargylformamide pesticides BAYER AKTIENGESELLSCHAFT (DE) 1987-04-28 US disclosed
EP-0094539-B1 HALOGENOPROPARGYL FORMAMIDES BAYER AG (DE) 1985-08-21 EP disclosed
EP-0094539-A1 Halogenopropargyl formamides BAYER AG (DE) 1983-11-23 EP disclosed