SCHEMBL794253

SCHEMBL794253

CC(C)(C)OC(=O)N[C@@H]1CCN(c2nc(N)nc3sc(-c4ccc(F)cc4)cc23)C1.Nc1nc(N2CCN(CCOc3ccccc3)CC2)c2cc(-c3ccccc3)sc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.43
HTR7 P34969 5/20 0.40
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39
SKP2 Q13309 1/20 0.39
AURKA O14965 3/20 0.39
PDPK1 O15530 3/20 0.39
AURKB Q96GD4 3/20 0.39
CNR2 P34972 4/20 0.38
CNR1 P21554 2/20 0.38
CYP2D6 P10635 1/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
PDE10A Q9Y233 1/20 0.38
HTR1A P08908 2/20 0.37
DRD2 P14416 1/20 0.37
HTR6 P50406 1/20 0.37
ALOX5AP P20292 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1721433 0.98 BTK (0.41) BTKHTR7CKS1BSKP1SKP2
SCHEMBL653783 0.87 AURKA (0.46) BTKAURKAPDPK1AURKBPDE10A
SCHEMBL653784 0.87 AURKA (0.46) BTKAURKAPDPK1AURKBPDE10A
SCHEMBL656583 0.86 CKS1B (0.49) BTKCKS1BSKP1SKP2AURKA
SCHEMBL656582 0.86 CKS1B (0.49) BTKCKS1BSKP1SKP2AURKA
SCHEMBL653066 0.79 CNR2 (0.55) AURKACNR2CNR1CYP2D6KDM4E
SCHEMBL794422 0.78 HRH4 (0.46) CNR2CNR1KDM4EMEN1KMT2A
SCHEMBL652168 0.75 ATF4 (0.43) ALDH1A1
SCHEMBL652167 0.75 ATF4 (0.43) ALDH1A1
SCHEMBL1694112 0.75 CNR2 (0.55) HTR7AURKACNR2CNR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011147753-A1 ANTIVIRAL ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2011-12-01 WO disclosed