SCHEMBL794422

SCHEMBL794422

Nc1nc(N2CCC(NC(=O)O)C2)c2cc(-c3ccc(F)cc3)sc2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 8/20 0.46
CNR2 P34972 3/20 0.43
PPARD Q03181 1/20 0.42
PPARA Q07869 1/20 0.42
SMPD3 Q9NY59 1/20 0.41
ACKR3 P25106 2/20 0.40
PIK3CA P42336 2/20 0.40
GRIA1 P42261 2/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
CNR1 P21554 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HRH3 Q9Y5N1 2/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653994 0.87 DRD2 (0.44) HRH4CNR2PPARDPPARACNR1
SCHEMBL653784 0.87 AURKA (0.46) HRH4
SCHEMBL653993 0.87 DRD2 (0.44) HRH4CNR2PPARDPPARACNR1
SCHEMBL653783 0.87 AURKA (0.46) HRH4
SCHEMBL652168 0.83 ATF4 (0.43) HRH4ALDH1A1LMNA
SCHEMBL652167 0.83 ATF4 (0.43) HRH4ALDH1A1LMNA
SCHEMBL655343 0.82 HRH4 (0.64) HRH4CNR2KDM4EALDH1A1MEN1
SCHEMBL655344 0.82 HRH4 (0.64) HRH4CNR2KDM4EALDH1A1MEN1
SCHEMBL1694133 0.80 HRH4 (0.45) HRH4ALDH1A1LMNA
SCHEMBL652787 0.80 DRD2 (0.46) HRH4CNR2PPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616077-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2013-07-24 EP claimed
WO-2012035423-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-03-22 WO claimed