SCHEMBL7944641

SCHEMBL7944641

N#Cc1cccc(-c2nc3c(N)ccnc3n(CC(F)(F)F)c2=O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 16/20 0.45
CYP1A2 P05177 14/20 0.45
USP2 O75604 14/20 0.45
HSD17B10 Q99714 12/20 0.45
CYP3A4 P08684 12/20 0.45
CASP1 P29466 12/20 0.45
CASP7 P55210 11/20 0.45
CYP2D6 P10635 6/20 0.45
MEN1 O00255 5/20 0.45
KMT2A Q03164 5/20 0.45
CLK4 Q9HAZ1 3/20 0.45
GLA P06280 2/20 0.45
HPGD P15428 3/20 0.45
HIF1A Q16665 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
CYP2C9 P11712 10/20 0.44
MAPK1 P28482 5/20 0.44
CFTR P13569 1/20 0.44
TSHR P16473 3/20 0.43
BLM P54132 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7938050 0.90 ALDH1A1 (0.47) ALDH1A1CYP1A2USP2HSD17B10CYP3A4
SCHEMBL7946753 0.85 ALDH1A1 (0.52) ALDH1A1CYP1A2USP2HSD17B10CYP3A4
SCHEMBL7938164 0.85 PDE4B (0.42) CLK4
SCHEMBL7949559 0.83 ALDH1A1 (0.49) ALDH1A1CYP1A2USP2HSD17B10CYP3A4
SCHEMBL7945959 0.83 PDE4B (0.51) ALDH1A1CYP1A2USP2HSD17B10CYP3A4
SCHEMBL7938295 0.83 ALDH1A1 (0.48) ALDH1A1CYP1A2USP2HSD17B10CYP3A4
SCHEMBL7944785 0.83 ALDH1A1 (0.47) ALDH1A1CYP1A2USP2HSD17B10CYP3A4
SCHEMBL7944623 0.83 ALDH1A1 (0.66) ALDH1A1CYP1A2USP2HSD17B10CYP3A4
SCHEMBL7938047 0.81 CYP1A2 (0.56) ALDH1A1CYP1A2USP2HSD17B10CYP3A4
SCHEMBL7945962 0.81 CYP1A2 (0.59) ALDH1A1CYP1A2USP2HSD17B10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed