SCHEMBL7945372

SCHEMBL7945372

CCOC(=O)c1cnc(N2CC3C2CN3C(c2ccccc2)c2ccccc2)nc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.43
OPRD1 P41143 1/20 0.41
P2RY12 Q9H244 6/20 0.40
OGA O60502 1/20 0.39
CACNA1A O00555 1/20 0.39
CACNA2D1 P54289 1/20 0.39
CACNB1 Q02641 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
GABRA1 P14867 2/20 0.39
GABRB2 P47870 2/20 0.39
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
LMNA P02545 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ABCB11 O95342 1/20 0.39
GABRA2 P47869 1/20 0.39
ALDH1A1 P00352 3/20 0.38
GAA P10253 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16302007 1.00 ACACB (0.43) ACACBOPRD1P2RY12OGACACNA1A
SCHEMBL1367800 0.83 ACACB (0.44) ACACBOPRD1P2RY12OGACACNA1A
SCHEMBL16302028 0.80 HDAC6 (0.49)
SCHEMBL12428624 0.71 ALDH1A1 (0.43) ACACBALDH1A1GAAMAPT
SCHEMBL7959667 0.71 ALDH1A1 (0.43) ACACBALDH1A1GAAMAPT
SCHEMBL1365631 0.70 CHRNB2 (0.46) ACACB
SCHEMBL21640616 0.70 OGA (0.49) OPRD1P2RY12OGACACNA1ACACNA2D1
SCHEMBL13535016 0.70 TSHR (0.62) P2RY12OGAALDH1A1GAAKDM4E
SCHEMBL16302029 0.68 ACACB (0.42) ACACBP2RY12OGACYP2C9CYP2C19
SCHEMBL9212828 0.67 P2RY12 (0.64) OPRD1P2RY12OGAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137503-A1 HDAC INHIBITORS AND USES THEREOF ENVIVO PHARMACEUTICALS, INC. (US) 2009-11-12 WO disclosed
WO-2009137462-A2 METHODS FOR TREATING COGNITIVE DISORDERS USING INHIBITORS OF HISTONE DEACETYLASE ENVIVO PHARMACEUTICALS, INC. (US) 2009-11-12 WO disclosed
WO-2008055068-A2 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2008-05-08 WO disclosed