SCHEMBL7945642

SCHEMBL7945642

Cc1ccc(Oc2cc[c]cn2)c(C)n1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 1/20 0.38
TGFBR1 P36897 4/20 0.35
GPR119 Q8TDV5 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5361562 0.79 MAP4K4 (0.44)
SCHEMBL7954135 0.75 GAA (0.43) S1PR4MEN1KMT2A
SCHEMBL2900836 0.75 HTT (0.37)
SCHEMBL2897755 0.75 SMN1; SMN2 (0.55) MEN1KMT2A
SCHEMBL7955819 0.73 SLC6A4 (0.45) MEN1KMT2A
SCHEMBL10393866 0.73 KDM4E (0.36) MEN1KMT2A
SCHEMBL2897754 0.71 MAP4K4 (0.43) TGFBR1KMT2A
SCHEMBL693585 0.71 KMT2A (0.49) MEN1KMT2A
SCHEMBL2894972 0.70 MEN1 (0.52) MEN1KMT2A
SCHEMBL2901162 0.70 SLC6A2 (0.32) S1PR4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235758-B1 CENTRAL NERVOUS SYSTEM DISORDERS SMITHKLINE BEECHAM P.L.C. (GB) 2001-05-22 US disclosed
EP-0808312-B1 INDOLE DERIVATIVES AS 5-HT RECEPTOR ANTAGONIST SMITHKLINE BEECHAM PLC (GB) 2000-11-02 EP disclosed
US-5990133-A TREATING CENTRAL NERVOUS SYSTEM DISORDERS SUCH AS ANXIETY OR DEPRESSION SMITHKLINE BEECHAM P.L.C. (GB) 1999-11-23 US disclosed