SCHEMBL7945757

SCHEMBL7945757

CC(C)[C@H](C#N)c1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.47
ESR2 Q92731 4/20 0.47
ADRB2 P07550 1/20 0.46
ALDH1A1 P00352 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 1/20 0.39
FFAR2 O15552 2/20 0.39
TSHR P16473 2/20 0.38
MAPK1 P28482 2/20 0.38
HIF1A Q16665 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
LMNA P02545 2/20 0.37
TP53 P04637 1/20 0.37
HPGD P15428 1/20 0.37
MAPT P10636 1/20 0.37
AOC3 Q16853 1/20 0.36
BRD4 O60885 1/20 0.35
CYP2A6 P11509 1/20 0.35
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2920989 1.00 ESR1 (0.47) ESR1ESR2ADRB2ALDH1A1L3MBTL1
SCHEMBL7939324 1.00 ESR1 (0.47) ESR1ESR2ADRB2ALDH1A1L3MBTL1
SCHEMBL1095072 0.83 ESR1 (0.48) ESR1ESR2ADRB2ALDH1A1L3MBTL1
SCHEMBL11229208 0.80 GAA (0.42) ESR1ESR2ADRB2ALDH1A1L3MBTL1
SCHEMBL9419163 0.78 ADRB2 (0.46) ADRB2GAAFFAR2TSHRMAPK1
SCHEMBL10952365 0.78 ESR1 (0.47) ESR1ESR2ALDH1A1GAAHPGD
SCHEMBL10706998 0.78 ESR1 (0.75) ESR1ESR2ALDH1A1TDP1LMNA
SCHEMBL7967104 0.78 ESR1 (0.47) ESR1ESR2ALDH1A1TDP1LMNA
SCHEMBL11070316 0.78 SLC6A3 (0.47) ESR1ESR2ALDH1A1LMNAIDO1
SCHEMBL10573002 0.77 SLC6A3 (0.41) ESR1ESR2ADRB2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251650-B1 Pseudomonas putida amidase polypeptide useful for the production of chiral amides and acids E. I. DU PONT DE NEMOURS AND COMPANY 2001-06-26 US disclosed
US-6133421-A FOR PRODUCTION OF AGROCHEMICALS AND PHARMACEUTICALS E. I. DU PONT DE NEMOURS & COMPANY (US) 2000-10-17 US disclosed
US-5888785-A USING NUCLEIC ACID ISOLATED FROM PEUDOMONAS AS CATALYST E. I. DU PONT DE NEMOURS AND COMPANY (US) 1999-03-30 US disclosed
US-5811286-A Nucleic acid fragments encoding stereospecific nitrile hydratase and amidase enzymes and recombinant organisms expressing those enzymes useful for the production of chiral amides and acids E. I. DU PONT DE NEMOURS AND COMPANY (US) 1998-09-22 US disclosed
EP-0853663-A1 NUCLEIC ACID FRAGMENTS ENCODING STEREOSPECIFIC NITRILE HYDRATASE AND AMIDASE ENZYMES AND RECOMBINANT MICROORGANISMS EXPRESSING THOSE ENZYMES USEFUL FOR THE PRODUCTION OF CHIRAL AMIDES AND ACIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-07-22 EP disclosed
WO-1997012964-A2 NUCLEIC ACID FRAGMENTS ENCODING STEREOSPECIFIC NITRILE HYDRATASE AND AMIDASE ENZYMES AND RECOMBINANT MICROORGANISMS EXPRESSING THOSE ENZYMES USEFUL FOR THE PRODUCTION OF CHIRAL AMIDES AND ACIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1997-04-10 WO disclosed