SCHEMBL7946501

SCHEMBL7946501

Bc1cc(C(=O)NCc2cnc(C)nc2)cc(-c2ccc(C)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.53
AKR1C3 P42330 12/20 0.50
AKR1C4 P17516 7/20 0.50
AKR1C2 P52895 6/20 0.50
AKR1C1 Q04828 2/20 0.50
P2RX3 P56373 2/20 0.48
P2RX2 Q9UBL9 2/20 0.48
KDM1A O60341 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1495662 0.91 AKR1C3 (0.55) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1
SCHEMBL1495539 0.87 AKR1C3 (0.54) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1
SCHEMBL2383698 0.86 AKR1C3 (0.53) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1
SCHEMBL2173876 0.85 P2RX3 (0.50) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1
SCHEMBL2170971 0.84 P2RX3 (0.67) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1
SCHEMBL12757591 0.83 AKR1C3 (0.56) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1
SCHEMBL28814525 0.83 AKR1C3 (0.47) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1
SCHEMBL1495717 0.83 AKR1C3 (0.50) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1
SCHEMBL1495365 0.83 AKR1C3 (0.49) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1
SCHEMBL1495558 0.82 AKR1C3 (0.49) HDAC1AKR1C3AKR1C4AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010033168-A2 AMIDE COMPOUNDS, COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2010-03-25 WO disclosed