SCHEMBL28814525

SCHEMBL28814525

Cc1ccc(-c2cc(C[SH](=O)=O)cc(C(=O)NCc3cnc(C)nc3)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 11/20 0.47
AKR1C4 P17516 7/20 0.47
AKR1C2 P52895 6/20 0.47
HDAC1 Q13547 3/20 0.47
AKR1C1 Q04828 2/20 0.47
P2RX3 P56373 2/20 0.46
P2RX2 Q9UBL9 2/20 0.46
WDR5 P61964 2/20 0.43
KDM1A O60341 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27981584 0.89 WDR5 (0.55) AKR1C3AKR1C4AKR1C2HDAC1AKR1C1
SCHEMBL1495662 0.88 AKR1C3 (0.55) AKR1C3AKR1C4AKR1C2HDAC1AKR1C1
SCHEMBL27981587 0.85 AKR1C3 (0.48) AKR1C3AKR1C4AKR1C2HDAC1AKR1C1
SCHEMBL2173876 0.84 P2RX3 (0.50) AKR1C3AKR1C4AKR1C2HDAC1AKR1C1
SCHEMBL1495539 0.84 AKR1C3 (0.54) AKR1C3AKR1C4AKR1C2HDAC1AKR1C1
SCHEMBL7946501 0.83 HDAC1 (0.53) AKR1C3AKR1C4AKR1C2HDAC1AKR1C1
SCHEMBL2383698 0.83 AKR1C3 (0.53) AKR1C3AKR1C4AKR1C2HDAC1AKR1C1
SCHEMBL27982185 0.82 P2RX3 (0.47) P2RX3P2RX2
SCHEMBL2170971 0.81 P2RX3 (0.67) AKR1C3AKR1C4AKR1C2HDAC1AKR1C1
SCHEMBL27981927 0.80 ROCK2 (0.40) P2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104058999-A Amide Compounds, Compositions And Uses Thereof RENOVIS INC 2014-09-24 CN disclosed
CN-104016907-A Amide compounds, compositions and uses thereof RENOVIS INC 2014-09-03 CN disclosed