SCHEMBL7946778

SCHEMBL7946778

O=C1CCOc2cc(OCc3ccccc3)c(F)cc21

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOB P27338 14/20 0.64
GRM5 P41594 9/20 0.64
NPC1 O15118 1/20 0.64
ALDH1A1 P00352 1/20 0.64
HPGD P15428 1/20 0.64
NFKB1 P19838 1/20 0.64
RAB9A P51151 1/20 0.64
NFKB2 Q00653 1/20 0.64
RELA Q04206 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
NPSR1 Q6W5P4 1/20 0.64
MAOA P21397 1/20 0.47
S1PR5 Q9H228 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30132495 0.85 MAOB (0.64) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL20554144 0.85 MAOB (0.64) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL27464278 0.81 MAOB (0.43) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL6836955 0.78 MAOB (0.81) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL2326572 0.78 MAOB (1.00) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL30353218 0.78 MAOB (0.81) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL29889798 0.78 MAOB (1.00) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL7940728 0.77 MAOB (0.42) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL20234906 0.77 MAOA (0.62) MAOBMAOA
SCHEMBL22712728 0.76 MAOB (0.62) MAOBGRM5NPC1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6258827-B1 HYDROXYAROMATIC HETEROCYCLIC ALKANOLS AND LEVODOPA PFIZER INC. 2001-07-10 US disclosed
US-6046213-A Neuroprotective 3-(piperidinyl-1)-chroman-4,7-diol and 1-(4-hydroxyphenyl)-2-(piperidinyl-1)-alkanol derivatives PFIZER INC. (US) 2000-04-04 US disclosed
EP-0828513-A2 COMBINATIONS FOR THE TREATMENT OF PARKINSONISM CONTAINING SELECTIVE NMDA ANTAGONISTS PFIZER INC. (US) 1998-03-18 EP disclosed
CN-1159325-A Co-therapy for Parkinson's syndrome PFIZER (US) 1997-09-17 CN disclosed
EP-0777652-A1 NEUROPROTECTIVE 3-(PIPERIDINYL-1)-CHROMAN-4,7-DIOL AND 1-(4-HYDROPHENYL)-2-(PIPERIDINYL-1)-ALKANOL DERIVATIVES PFIZER INC. (US) 1997-06-11 EP disclosed
WO-1996037226-A2 COMBINATIONS FOR THE TREATMENT OF PARKINSONISM CONTAINING SELECTIVE NMDA ANTAGONISTS PFIZER INC. (US) 1996-11-28 WO disclosed
WO-1996006081-A1 NEUROPROTECTIVE 3-(PIPERIDINYL-1)-CHROMAN-4,7-DIOL AND 1-(4-HYDROPHENYL)-2-(PIPERIDINYL-1)-ALKANOL DERIVATIVES PFIZER INC. (US) 1996-02-29 WO disclosed