SCHEMBL7947925

SCHEMBL7947925

Nc1ccnc2c1nc(-c1nccs1)c(=O)n2CC1CC1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 8/20 0.36
ADORA2A P29274 9/20 0.34
ADORA3 P0DMS8 4/20 0.34
PDE4B Q07343 5/20 0.33
PDE5A O76074 4/20 0.33
PDE4A P27815 4/20 0.33
PDE4C Q08493 4/20 0.33
PDE4D Q08499 4/20 0.33
ADORA2B P29275 4/20 0.33
HSP90AA1 P07900 1/20 0.33
CDC7 O00311 1/20 0.33
OPRD1 P41143 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7944078 0.82 PDE4B (0.42) ADORA1ADORA2AADORA3PDE4BADORA2B
SCHEMBL7947387 0.81 ADORA1 (0.36) ADORA1ADORA2AADORA3PDE4BADORA2B
SCHEMBL3227759 0.81 ALDH1A1 (0.39) ADORA1ADORA2AADORA3ADORA2BHSP90AA1
SCHEMBL7944114 0.80 PDE4B (0.48) ADORA1ADORA2AADORA3PDE4BPDE4A
SCHEMBL7947184 0.80 CYP1A2 (0.45)
SCHEMBL7946078 0.79 ADORA1 (0.36) ADORA1ADORA2AADORA3ADORA2BHSP90AA1
SCHEMBL7938177 0.78 PDE4B (0.41) ADORA2APDE4BPDE4APDE4CPDE4D
SCHEMBL7949559 0.74 ALDH1A1 (0.49) ADORA2A
SCHEMBL7946794 0.68 ADORA1 (0.39) ADORA1ADORA2AADORA3PDE4BADORA2B
SCHEMBL3227758 0.66 CYP1A2 (0.41) ADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed