SCHEMBL7948338

SCHEMBL7948338

NC(=O)CO[C@@H]1[C@H](O)[C@@H](Oc2ccc([N+](=O)[O-])cc2)O[C@H](COC(c2ccccc2)(c2ccccc2)c2ccccc2)[C@H]1O

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.39
HPSE Q9Y251 1/20 0.35
TYMP P19971 6/20 0.34
ALDH1A1 P00352 3/20 0.33
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7958047 0.90 NT5E (0.38) NT5EHPSETYMPALDH1A1SMN1; SMN2
SCHEMBL7948150 0.90 NT5E (0.38) NT5EHPSETYMPALDH1A1CYP2C9
SCHEMBL7955444 0.88 NT5E (0.50) NT5EHPSETYMP
SCHEMBL7955443 0.88 NT5E (0.50) NT5EHPSETYMP
SCHEMBL7958046 0.88 NT5E (0.44) NT5EHPSETYMPALDH1A1LMNA
SCHEMBL7957807 0.86 TYMP (0.38) NT5EHPSETYMPALDH1A1
SCHEMBL7962368 0.85 TYR (0.42) NT5EHPSETYMPALDH1A1
SCHEMBL7962363 0.85 TYR (0.42) NT5EHPSETYMPALDH1A1
SCHEMBL7948155 0.85 TYR (0.42) NT5EHPSETYMPALDH1A1
SCHEMBL7959227 0.83 CYP1A2 (0.45) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271342-B1 SERUM STABILITY; FOR TUMOR THERAPY BAYER AKTIENGESELLSCHAFT (DE) 2001-08-07 US disclosed
EP-0819135-B1 SUGAR-MODIFIED CYTOSTATICS BAYER AG (DE) 1999-11-17 EP disclosed
EP-0819135-A1 SUGAR-MODIFIED CYTOSTATICS BAYER AG (DE) 1998-01-21 EP disclosed
WO-1996031532-A1 SUGAR-MODIFIED CYTOSTATICS BAYER AKTIENGESELLSCHAFT (DE) 1996-10-10 WO disclosed