SCHEMBL7948821

SCHEMBL7948821

C#CC1CCc2ccccc2O1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.41
HTR1A P08908 6/20 0.39
SIGMAR1 Q99720 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
ADRA2A P08913 1/20 0.39
HTR1D P28221 4/20 0.37
MAOA P21397 4/20 0.36
MAOB P27338 4/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
ADRA1A P35348 1/20 0.36
HTR6 P50406 1/20 0.36
NISCH Q9Y2I1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5695479 0.81 CA2 (0.41) CA2HTR1ASIGMAR1ADRA2BADRA2C
SCHEMBL29644533 0.81 CA2 (0.41) CA2HTR1ASIGMAR1ADRA2BADRA2C
SCHEMBL4289906 0.81 CA2 (0.41) CA2HTR1ASIGMAR1ADRA2BADRA2C
SCHEMBL95677 0.81 CA2 (0.44) CA2HTR1ASIGMAR1ADRA2BADRA2C
SCHEMBL5130635 0.81 MAOB (0.38) MAOAMAOBNISCH
SCHEMBL460126 0.75 CA2 (0.44) CA2HTR1ASIGMAR1ADRA2BADRA2C
SCHEMBL30070640 0.75 CA2 (0.44) CA2HTR1ASIGMAR1ADRA2BADRA2C
SCHEMBL1567113 0.75 HTR1A (0.45) CA2HTR1ASIGMAR1ADRA2BADRA2C
SCHEMBL29462397 0.74 CA2 (0.46) CA2HTR1ASIGMAR1ADRA2BADRA2C
SCHEMBL9006852 0.74 ESR1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6258811-B1 ADMINISTERING RETINOIC ACID RECEPTOR AGONIST EISAI CO., LTD. (JP) 2001-07-10 US claimed
US-6258811-B1 ADMINISTERING RETINOIC ACID RECEPTOR AGONIST EISAI CO., LTD. (JP) 2001-07-10 US disclosed
EP-0930075-A1 METHODS FOR PREVENTING, INHIBITING OR TREATING GRAFT REJECTION REACTIONS IN GRAFT-VERSUS-HOST DISEASE (GVHD) AND ORGAN TRANSPLANTATION Eisai Co., Ltd. (JP) 1999-07-21 EP disclosed
EP-0320777-B1 A NOVEL APPROACH TO PRODUCE NATURAL VITAMIN E MAKING USE OF AN ASYMMETRIC SYNTHESIS F. HOFFMANN-LA ROCHE AG (CH) 1992-03-18 EP disclosed
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
EP-0320777-A2 A novel approach to produce natural vitamin E making use of an asymmetric synthesis F. HOFFMANN-LA ROCHE AG (CH) 1989-06-21 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed