SCHEMBL7950100

SCHEMBL7950100

COc1ccc2c(C(=O)c3ccc(OCCN4CCCC4)cc3)c(-c3ccc(OCCN4CCCC4)cc3)[s+]([O-])c2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 17/20 0.61
ESR2 Q92731 17/20 0.61
ENPP3 O14638 1/20 0.54
ENPP1 P22413 1/20 0.54
PSMB1 P20618 1/20 0.53
PSMB5 P28074 1/20 0.53
PSMB2 P49721 1/20 0.53
MEN1 O00255 1/20 0.51
PLD2 O14939 1/20 0.51
KDM1A O60341 1/20 0.51
NR1I2 O75469 1/20 0.51
USP2 O75604 1/20 0.51
ALDH1A1 P00352 1/20 0.51
C5 P01031 1/20 0.51
LMNA P02545 1/20 0.51
TP53 P04637 1/20 0.51
FYN P06241 1/20 0.51
PGR P06401 1/20 0.51
CYP3A4 P08684 1/20 0.51
ADRA2A P08913 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11551921 0.99 ESR1 (0.63) ESR1ESR2ENPP3ENPP1PSMB1
SCHEMBL11551029 0.96 ESR1 (0.66) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL11551801 0.96 ESR1 (0.59) ESR1ESR2ENPP3ENPP1PSMB1
SCHEMBL11555041 0.96 ESR1 (0.66) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL11553642 0.95 ESR1 (0.56) ESR1ESR2ENPP3ENPP1DRD3
SCHEMBL11546606 0.95 ESR1 (0.56) ESR1ESR2ENPP3ENPP1PSMB1
SCHEMBL11549231 0.92 PSMB1 (0.52) ESR1ESR2ENPP3PSMB1PSMB5
SCHEMBL7775848 0.90 ESR1 (0.62) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL11548378 0.89 ESR1 (0.64) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL8920012 0.88 ESR1 (0.64) ESR1ESR2MEN1PLD2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed