SCHEMBL7950125

SCHEMBL7950125

COc1ccc2c(c1)C(CCNC(=O)C(F)(F)F)C(C)(C)CC2

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 16/20 0.67
MTNR1B P49286 16/20 0.67
NQO2 P16083 16/20 0.67
ADRB2 P07550 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47
ADRA2B P18089 1/20 0.47
SLC6A2 P23975 1/20 0.47
HTR2C P28335 1/20 0.47
HRH1 P35367 1/20 0.47
OPRM1 P35372 1/20 0.47
OPRK1 P41145 1/20 0.47
HTR2B P41595 1/20 0.47
HTR5A P47898 1/20 0.47
SLC6A3 Q01959 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
TRPV1 Q8NER1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7943657 0.89 MTNR1A (0.64) MTNR1AMTNR1BNQO2
SCHEMBL7945323 0.87 MTNR1A (0.53) MTNR1AMTNR1BNQO2ADRB2HTR1A
SCHEMBL7953980 0.87 MTNR1A (0.65) MTNR1AMTNR1BNQO2ADRB2HTR1A
SCHEMBL7950253 0.85 MTNR1A (0.62) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL7954049 0.84 TRPV1 (0.55) MTNR1AMTNR1BNQO2ADRB2HTR1A
SCHEMBL7951392 0.81 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL7951348 0.81 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL7951573 0.81 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL7951212 0.79 MTNR1A (1.00) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL7950457 0.79 MTNR1A (1.00) MTNR1AMTNR1BNQO2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235789-B1 GLANDULAR DISORDERS; SLEEP DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0781271-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-07-02 EP disclosed
WO-1996008466-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-21 WO disclosed