SCHEMBL7950467

SCHEMBL7950467

COc1c(C)cnc(Cl)c1C

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AGXT P21549 1/20 0.50
HSP90AA1 P07900 18/20 0.42
HSP90AB1 P08238 10/20 0.42
TRAP1 Q12931 2/20 0.42
HSP90B1 P14625 1/20 0.42
ATP4A P20648 1/20 0.36
ATP4B P51164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL31097366 0.98 AGXT (0.49) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL26281215 0.84 AGXT (0.43) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1
Hydrochloric Acid SCHEMBL3180897 0.83 AGXT (0.42) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL94923 0.77 AGXT (0.53) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1
Hydrochloric Acid SCHEMBL28303939 0.76 AGXT (0.52) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL29039529 0.76 AGXT (0.52) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL29736023 0.76 AGXT (0.52) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL7845798 0.76 AGXT (0.52) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL22586637 0.75 AGXT (0.40) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL94922 0.74 AGXT (0.50) AGXTHSP90AA1HSP90AB1TRAP1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101906106-A New heterogeneous ring compound as the HSP90-inhibitor CONFORMA THERAPEUTICS CORP 2010-12-08 CN disclosed
CN-1882589-B Novel heterocyclic compounds as HSP 90-inhibitors CONFORMA THERAPEUTICS CORP 2010-06-09 CN disclosed
CN-1882589-A Novel heterocyclic compounds as HSP 90-inhibitors CONFORMA THERAPEUTICS CORP (US) 2006-12-20 CN disclosed
US-6303787-B1 STARTING FROM 4-NITRO-2,3,5-TRIMETHYLPYRIDINE-N-OXIDE AND5-METHOXY-2-MERCAPTO BENZIMIDAZOLE NATCO PHARMA LIMITED (IN) 2001-10-16 US disclosed
CN-85103357-A The method for making of tricyclic imidazole derivatives and acid salt thereof 1986-11-12 CN disclosed