SCHEMBL7950707

SCHEMBL7950707

Cc1ccc2c(c1)N(CC(=O)c1ccccc1C)C(=O)C(NC(=O)OC(C)(C)C)CN2C(=O)OCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.38
CCKBR P32239 4/20 0.38
MAPT P10636 2/20 0.37
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
CASP1 P29466 1/20 0.36
RORC P51449 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
NPY1R P25929 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6177392 0.88 CCKBR (0.39) CCKBRMAPTCYP3A4TSHRLMNA
SCHEMBL6177504 0.88 CCKBR (0.39) CCKBRMAPTCYP3A4TSHR
SCHEMBL6176603 0.87 CCKBR (0.39) CCKBRMAPTCYP3A4TSHRLMNA
SCHEMBL7959399 0.86 CCKBR (0.38) CCKBRMAPTCYP3A4TSHRLMNA
SCHEMBL7959563 0.86 HTT (0.37) CCKBRMAPTCYP3A4TSHRNPY1R
SCHEMBL6178660 0.85 CCKBR (0.38) CCKBRMAPTCYP3A4TSHRLMNA
SCHEMBL7950861 0.85 CCKBR (0.37) CCKBRMAPTCYP3A4TSHRNPY1R
SCHEMBL6176875 0.85 CCKBR (0.39) CCKBRMAPTCYP3A4TSHR
SCHEMBL7961009 0.84 CCKBR (0.38) CCKBRMAPTCYP3A4TSHR
SCHEMBL6176839 0.83 HTT (0.41) PDE4BLMNASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed