SCHEMBL7951247

SCHEMBL7951247

S=C1CN=C(c2ccccn2)c2cc(I)ccc2N1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 9/20 0.65
ADRA1A P35348 1/20 0.54
ALDH1A1 P00352 1/20 0.49
PKM P14618 1/20 0.49
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALOX12 P18054 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CCNB2 O95067 1/20 0.39
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
GABRA1 P14867 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35
GABRA2 P47869 2/20 0.35
GABRB2 P47870 2/20 0.35
CNR1 P21554 1/20 0.33
NTSR1 P30989 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374778 0.85 ADRA1A (0.74) CHRM1ADRA1AALDH1A1PKMHTT
SCHEMBL7376835 0.85 CHRM1 (0.69) CHRM1ADRA1AALDH1A1PKMHTT
SCHEMBL7951942 0.85 ADRA1A (0.74) CHRM1ADRA1AGABRA1GABRA5GABRA3
SCHEMBL11837472 0.85 ADRA1A (0.54) CHRM1ADRA1AALDH1A1PKMHTT
SCHEMBL11837680 0.84 ADRA1A (0.51) CHRM1ADRA1AALDH1A1PKMHTT
SCHEMBL11606414 0.82 CHRM1 (0.71) CHRM1ADRA1AALDH1A1PKMHTT
SCHEMBL11828237 0.82 CHRM1 (0.71) CHRM1ADRA1AALDH1A1PKMHTT
SCHEMBL10741591 0.82 CHRM1 (0.71) CHRM1ALDH1A1PKMHTTNPSR1
SCHEMBL11825591 0.80 CHRM1 (0.72) CHRM1ADRA1AALDH1A1PKMHTT
SCHEMBL7950385 0.79 CHRM1 (1.00) CHRM1ALDH1A1PKMHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174881-B1 USED AS ANXIOLYTIC AND/OR ANTICONVULSANT AND/OR MUSCLE RELAXANT AGENTS; SEDATIVES OR HYPNOSIS; WATER-SOLUBLE AMINE SALTS; FAST-ACTING HOFFMAN-LA ROCHE INC. 2001-01-16 US disclosed