SCHEMBL795138

SCHEMBL795138

Nc1nc(N2CCNCC2C(=O)CCc2ccccc2)c2cc(-c3ccc(F)cc3)sc2n1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 2/20 0.36
SCN9A Q15858 2/20 0.36
USP25 Q9UHP3 4/20 0.35
USP28 Q96RU2 2/20 0.35
HRH4 Q9H3N8 3/20 0.35
CNR2 P34972 2/20 0.35
HRH3 Q9Y5N1 1/20 0.35
GPR55 Q9Y2T6 1/20 0.34
CHEK1 O14757 3/20 0.34
KCNH2 Q12809 1/20 0.34
LSS P48449 1/20 0.33
KIT P10721 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
GRM2 Q14416 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12467234 0.82 CHEK1 (0.39) FPR2SCN9AHRH4HRH3CHEK1
SCHEMBL1693574 0.82 FPR2 (0.39) FPR2SCN9AHRH4HRH3CHEK1
SCHEMBL1694252 0.81 CYP1A2 (0.37) FPR2SCN9ACHEK1KCNH2LSS
SCHEMBL656257 0.78 GFER (0.53) CNR2GPR55KIT
SCHEMBL653761 0.75 HRH4 (0.41) FPR2SCN9AHRH4HRH3CHEK1
SCHEMBL655042 0.72 HRH4 (0.61) HRH4CNR2HRH3KCNH2
SCHEMBL660185 0.70 CYP2D6 (0.41) HRH4CNR2
SCHEMBL653372 0.70 CNR2 (0.48) HRH4CNR2GPR55
SCHEMBL4778347 0.69 HRH4 (0.43) FPR2SCN9AHRH4HRH3KCNH2
SCHEMBL653760 0.69 KDM4E (0.50) HRH4CNR2GPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616077-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2013-07-24 EP disclosed
EP-2575969-A1 ANTIVIRAL ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2013-04-10 EP disclosed
WO-2012035423-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-03-22 WO disclosed