SCHEMBL7952022

SCHEMBL7952022

Clc1cc2nc(-c3ccccn3)c(-c3ccccn3)nc2cc1Cl

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.70
NPC1 O15118 3/20 0.70
CCR1 P32246 3/20 0.53
CCR5 P51681 3/20 0.53
CCR8 P51685 3/20 0.53
ADORA2A P29274 1/20 0.49
ADORA1 P30542 1/20 0.49
METAP1 P53582 3/20 0.48
LMNA P02545 2/20 0.48
CYP1A2 P05177 1/20 0.48
POLB P06746 1/20 0.48
BLM P54132 1/20 0.48
HIF1A Q16665 1/20 0.48
DOHH Q9BU89 1/20 0.48
P4HTM Q9NXG6 1/20 0.48
TP53 P04637 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
MAPK1 P28482 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7236265 0.91 KDM4E (0.59) KDM4ENPC1CCR1CCR5CCR8
SCHEMBL7965339 0.88 KDM4E (0.81) KDM4ENPC1CCR1CCR5CCR8
SCHEMBL7963689 0.84 KDM4E (0.75) KDM4ENPC1CCR1CCR5CCR8
SCHEMBL4075083 0.82 KDM4E (1.00) KDM4ENPC1CCR1CCR5CCR8
SCHEMBL2061612 0.81 KDM4E (0.70) KDM4ENPC1CCR1CCR5CCR8
SCHEMBL27928516 0.81 KDM4E (0.70) KDM4ENPC1CCR1CCR5CCR8
SCHEMBL7952005 0.79 KDM4E (0.68) KDM4ENPC1CCR1CCR5CCR8
SCHEMBL323086 0.79 KDM4E (0.68) KDM4ENPC1CCR1CCR5CCR8
SCHEMBL14063447 0.78 KDM4E (0.66) KDM4ENPC1CCR1CCR5CCR8
SCHEMBL21941944 0.77 METAP1 (0.57) KDM4ENPC1CCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187928-B1 TREATING FUNGAL DISEASES THE ROCKEFELLER UNIVERSITY 2001-02-13 US disclosed
US-6087510-A Method of use of imidazolium cations THE ROCKEFELLER UNIVERSITY (US) 2000-07-11 US disclosed
US-5969150-A FLUORESCENT COMPOUNDS FOR MEDICAL DIAGNOSIS, DRUGS AND LABELS OR FUNGICIDES AND VIRICIDES THE ROCKEFELLER UNIVERSITY (US) 1999-10-19 US disclosed
US-5874587-A FLUORESCENCE THE ROCKEFELLER UNIVERSITY (US) 1999-02-23 US disclosed