SCHEMBL7952134

SCHEMBL7952134

CC(C)Oc1ccc2c(c1)C(=CCNC(=O)C(F)(F)F)CCCC2

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 12/20 0.49
MTNR1B P49286 12/20 0.49
NQO2 P16083 12/20 0.49
THRB P10828 1/20 0.36
ADCY8 P40145 1/20 0.35
ADCY1 Q08828 1/20 0.35
PDK2 Q15119 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
CES2 O00748 1/20 0.34
ABCB1 P08183 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7952132 1.00 MTNR1A (0.49) MTNR1AMTNR1BNQO2THRBADCY8
SCHEMBL7952097 0.89 MTNR1A (0.62) MTNR1AMTNR1BNQO2ABCB1
SCHEMBL7952100 0.89 MTNR1A (0.62) MTNR1AMTNR1BNQO2ABCB1
SCHEMBL7952090 0.87 MTNR1A (0.62) MTNR1AMTNR1BNQO2ABCB1
SCHEMBL7952086 0.87 MTNR1A (0.62) MTNR1AMTNR1BNQO2ABCB1
SCHEMBL7952088 0.87 MTNR1A (0.62) MTNR1AMTNR1BNQO2ABCB1
SCHEMBL7951379 0.87 MTNR1A (0.53) MTNR1AMTNR1BNQO2THRBADCY8
SCHEMBL7951378 0.87 MTNR1A (0.53) MTNR1AMTNR1BNQO2THRBADCY8
SCHEMBL7945336 0.82 MTNR1A (0.71) MTNR1AMTNR1BNQO2
SCHEMBL7945340 0.82 MTNR1A (0.71) MTNR1AMTNR1BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235789-B1 GLANDULAR DISORDERS; SLEEP DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0781271-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-07-02 EP disclosed
WO-1996008466-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-21 WO disclosed