SCHEMBL7953183

SCHEMBL7953183

COc1ccc(CN(Cc2ccc(OC)cc2)c2ncnc3cncnc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
LMNA P02545 4/20 0.42
MAPT P10636 2/20 0.42
EGFR P00533 4/20 0.41
NOS1 P29475 1/20 0.39
MEN1 O00255 3/20 0.39
TSHR P16473 3/20 0.39
KMT2A Q03164 3/20 0.39
CYP3A4 P08684 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CHRM2 P08172 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
DRD1 P21728 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
SLC6A4 P31645 1/20 0.39
CYP2C19 P33261 1/20 0.39
HRH1 P35367 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL168410 0.82 KDM4E (0.49) ALDH1A1LMNAMAPTEGFRNOS1
SCHEMBL29809031 0.80 ALDH1A1 (0.46) ALDH1A1LMNAMAPTEGFRNOS1
SCHEMBL30949914 0.77 LMNA (0.43) ALDH1A1LMNAMAPTNOS1MEN1
SCHEMBL30949966 0.76 LMNA (0.42) ALDH1A1LMNAMAPTEGFRNOS1
SCHEMBL14574648 0.76 ALDH1A1 (0.41) ALDH1A1LMNAMAPTEGFRNOS1
Hydrochloric Acid SCHEMBL31152319 0.73 LMNA (0.41) ALDH1A1LMNAMAPTNOS1MEN1
SCHEMBL12825893 0.72 PTPN1 (0.42) ALDH1A1LMNAMAPTNOS1TSHR
SCHEMBL1461757 0.72 AURKA (0.42) ALDH1A1LMNAMAPTEGFRMEN1
SCHEMBL8132510 0.71 LMNA (0.53) ALDH1A1LMNAEGFRTSHRSMN1; SMN2
SCHEMBL30950103 0.71 ALDH1A1 (0.39) ALDH1A1LMNAMAPTMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2001517226-A 2001-10-02 JP claimed
EP-0971925-A1 PYRIMIDOPYRIMIDINE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 2000-01-19 EP claimed
WO-1998043974-A1 PYRIMIDOPYRIMIDINE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 1998-10-08 WO claimed