SCHEMBL7954276

SCHEMBL7954276

NC(=O)C1COCCN1C(=O)CN1CCNCC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
HSD17B10 Q99714 2/20 0.38
TSHR P16473 2/20 0.38
ALOX15 P16050 1/20 0.38
SIGMAR1 Q99720 4/20 0.35
CHRM5 P08912 2/20 0.35
CHRM3 P20309 2/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
SMYD3 Q9H7B4 2/20 0.33
FKBP1A P62942 1/20 0.33
GAA P10253 1/20 0.32
LMNA P02545 1/20 0.31
RAB9A P51151 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28310283 0.73 CA12 (0.45) KDM4ECA12CA1CA2CA9
SCHEMBL29022309 0.72 CA12 (0.44) KDM4EHSD17B10CA12CA1CA2
SCHEMBL1150296 0.72 CA12 (0.44) KDM4EHSD17B10CA12CA1CA2
SCHEMBL255444 0.71 HSD17B10 (0.69) KDM4EHSD17B10TSHRALOX15GAA
SCHEMBL2073211 0.71 HSD17B10 (0.69) KDM4EHSD17B10TSHRALOX15GAA
Hydrochloric Acid SCHEMBL1156139 0.69 HSD17B10 (0.67) KDM4EHSD17B10TSHRALOX15GAA
SCHEMBL4140585 0.69 L3MBTL1 (0.37) KDM4EHSD17B10TSHRALOX15CA12
SCHEMBL13893263 0.68 HSD17B10 (0.65) KDM4EHSD17B10TSHRALOX15GAA
SCHEMBL4087862 0.68 CA12 (0.41) KDM4ECA12CA1CA2CA9
SCHEMBL4163105 0.68 CA12 (0.41) KDM4ECA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6258815-B1 HETEROCYCLIC COMPOUNDS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 2001-07-10 US claimed
US-6258815-B1 HETEROCYCLIC COMPOUNDS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 2001-07-10 US disclosed