SCHEMBL7954544

SCHEMBL7954544

CCCCCCCCCC(Br)Oc1ccc(C2c3ccc(OCc4ccccc4)cc3OCC2c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.44
ESR2 Q92731 5/20 0.44
CTRC Q99895 1/20 0.38
HTR2B P41595 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
FFAR1 O14842 5/20 0.38
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
CA2 P00918 1/20 0.37
CA5A P35218 1/20 0.37
MAOB P27338 3/20 0.37
MAOA P21397 2/20 0.37
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6898886 0.88 ESR1 (0.43) ESR1ESR2CTRCHTR2BTMEM97
SCHEMBL6895273 0.85 ESR1 (0.44) ESR1ESR2CTRCHTR2BTMEM97
SCHEMBL6901793 0.83 ESR1 (0.44) ESR1ESR2HTR2BTMEM97SIGMAR1
SCHEMBL7056046 0.80 ESR1 (0.51) ESR1ESR2HTR2BTMEM97SIGMAR1
SCHEMBL6895957 0.80 ESR1 (0.62) ESR1ESR2HTR2BTMEM97SIGMAR1
SCHEMBL6900049 0.79 ESR1 (0.55) ESR1ESR2HTR2BTMEM97SIGMAR1
SCHEMBL6901973 0.79 ESR1 (0.55) ESR1ESR2HTR2BTMEM97SIGMAR1
SCHEMBL6899567 0.79 ESR1 (0.46) ESR1ESR2HTR2BTMEM97SIGMAR1
SCHEMBL6901788 0.79 ESR1 (0.51) ESR1ESR2HTR2BTMEM97SIGMAR1
SCHEMBL6901001 0.79 ESR1 (0.51) ESR1ESR2HTR2BTMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316494-B1 FOR THERAPY AND PROPHYLAXIS OF BONE LOSS, OSTEOPOROSIS, CARDIOVASCULAR DISEASES, COGNITIVE DISORDERS, MENOPAUSAL SYMPTOMS, INCONTINENCE, OBESITY, DYSMENORRHEA, DYSFUNCTIONAL UTERINE BLEEDING, ACNE, HIRSUTISM, POST-PARTUM LACTATION NOVO NORDISK A/S (DK) 2001-11-13 US disclosed