SCHEMBL7955355

SCHEMBL7955355

NC(=O)C(O)c1cccs1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.61
CES1 P23141 2/20 0.61
KEAP1 Q14145 1/20 0.61
ALOX5 P09917 2/20 0.51
ALDH1A1 P00352 3/20 0.40
MAPT P10636 3/20 0.40
HPGD P15428 2/20 0.40
PKM P14618 1/20 0.40
HTT P42858 1/20 0.40
ATM Q13315 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TSHR P16473 1/20 0.40
POLB P06746 3/20 0.39
CHRM3 P20309 1/20 0.39
DAO P14920 1/20 0.39
CYP2C19 P33261 1/20 0.37
MAPK10 P53779 1/20 0.37
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12238428 0.81 CES2 (0.63) CES2CES1KEAP1ALOX5ALDH1A1
SCHEMBL12238427 0.81 CES2 (0.63) CES2CES1KEAP1ALOX5ALDH1A1
SCHEMBL11077401 0.81 CES2 (0.63) CES2CES1KEAP1ALOX5ALDH1A1
SCHEMBL2547968 0.81 CES2 (0.63) CES2CES1KEAP1ALOX5ALDH1A1
SCHEMBL18824383 0.79 CES2 (0.52) CES2CES1KEAP1ALOX5ALDH1A1
SCHEMBL14828713 0.79 CES2 (0.61) CES2CES1KEAP1ALOX5ALDH1A1
SCHEMBL13163250 0.79 ALOX5 (0.51) CES2CES1KEAP1ALOX5ALDH1A1
SCHEMBL5027606 0.79 ALOX5 (0.51) CES2CES1KEAP1ALOX5ALDH1A1
SCHEMBL602500 0.78 ALOX5 (0.50) CES2CES1KEAP1ALOX5ALDH1A1
SCHEMBL8853390 0.78 ALOX5 (0.50) CES2CES1KEAP1ALOX5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4407815-A AMINO ACID DERIVATIVE ANTIBIOTICS BEECHAM GROUP LIMITED (GB) 1983-10-04 US claimed
US-6265519-B1 CURING AN EPOXIDE MOLEX INCORPORATED 2001-07-24 US disclosed
EP-0034443-B1 BETA-LACTAM ANTIBACTERIAL COMPOUNDS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1984-09-26 EP disclosed
US-4407815-A AMINO ACID DERIVATIVE ANTIBIOTICS BEECHAM GROUP LIMITED (GB) 1983-10-04 US disclosed
US-4387051-A β-Lactam antibiotics, their preparation and their use in pharmaceutical compositions BEECHAM GROUP LIMITED (GB) 1983-06-07 US disclosed
EP-0073100-A1 Beta-lactam compounds, their preparation and their use BEECHAM GROUP PLC (GB) 1983-03-02 EP disclosed
US-4329454-A Cephalosporin compounds ELI LILLY AND COMPANY (US) 1982-05-11 US disclosed
EP-0034443-A2 Beta-lactam antibacterial compounds, their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1981-08-26 EP disclosed
EP-0028497-A1 Beta-lactam antibiotics, their preparation and their use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-05-13 EP disclosed
US-4144391-A REPLACING AN ACETOXY GROUP BY A SULFUR NUCLEOPHILE ELI LILLY AND COMPANY (US) 1979-03-13 US disclosed