SCHEMBL7955384

SCHEMBL7955384

O=C(Nc1c(Cl)cccc1Cl)c1cn([C@H]2CCN(C(=O)OCc3ccccc3)C2)c2ncccc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.44
KCNH2 Q12809 2/20 0.44
GRIN2B Q13224 7/20 0.42
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
HTR6 P50406 1/20 0.39
CYP2C19 P33261 1/20 0.39
USP30 Q70CQ3 1/20 0.39
CYP2D6 P10635 4/20 0.38
CYP2C9 P11712 4/20 0.38
CYP3A4 P08684 3/20 0.38
ENPP2 Q13822 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7955386 1.00 PDE4A (0.44) PDE4AKCNH2GRIN2BSMN1; SMN2NPC1
SCHEMBL7953478 0.94 PDE4A (0.53) PDE4AKCNH2GRIN2BSMN1; SMN2NPC1
SCHEMBL7953479 0.94 PDE4A (0.53) PDE4AKCNH2GRIN2BSMN1; SMN2NPC1
SCHEMBL7960495 0.89 PDE4A (0.54) PDE4AKCNH2GRIN2BSMN1; SMN2NPC1
SCHEMBL7954854 0.88 KCNH2 (0.47) PDE4AKCNH2HTR6CYP2C19CYP2C9
SCHEMBL7953511 0.88 KCNH2 (0.47) PDE4AKCNH2HTR6CYP2C19CYP2C9
SCHEMBL7960298 0.88 KCNH2 (0.47) PDE4AKCNH2HTR6CYP2C19CYP2C9
SCHEMBL7954726 0.87 GRIN2B (0.46) GRIN2BSMN1; SMN2NPC1RAB9AHTR6
SCHEMBL7954870 0.87 GRIN2B (0.46) GRIN2BSMN1; SMN2NPC1RAB9AHTR6
SCHEMBL7963486 0.82 GRIN2B (0.50) GRIN2BSMN1; SMN2NPC1RAB9ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6331548-B1 PREVENTION OR TREATMENT OF CYTOKINE RELATED DISEASES SUNTORY LIMITED (JP) 2001-12-18 US disclosed
EP-0978516-A1 1-CYCLOALKYL-1,8-NAPHTHYRIDIN-4-ONE DERIVATIVES WITH PHOSPHODIESTERASE IV INHIBITORY ACTIVITY SUNTORY LIMITED (JP) 2000-02-09 EP disclosed