SCHEMBL7956727

SCHEMBL7956727

COc1ccc(S(=O)(=O)N(CC(C)C)C[C@@H](O)COC(=O)NCc2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.54
TP53 P04637 1/20 0.52
BACE1 P56817 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2582390 0.83 BACE1 (0.52) CXCR3BACE1
SCHEMBL4911761 0.82 CXCR3 (0.52) CXCR3
SCHEMBL14647093 0.79 BACE1 (0.58) CXCR3BACE1
SCHEMBL8436783 0.77 TP53 (0.64) CXCR3TP53
SCHEMBL12621038 0.75 SPPL2A (0.54)
SCHEMBL9287153 0.75 RORC (0.68) CXCR3BACE1
SCHEMBL11988980 0.75 SPPL2A (0.75)
SCHEMBL1804868 0.74 SPPL2A (0.60)
SCHEMBL6099960 0.74 SPPL2A (0.60)
SCHEMBL1804866 0.74 SPPL2A (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6169085-B1 A VIRICIDE FOR PREVENTING AND TREATING RETROVIRAL INFECTION OR THE SPREAD OF A RETROVIRUS, INHIBITING REPLICATION OF A RETROVIRUS AND TREATING AIDS G. D. SEARLE & COMPANY 2001-01-02 US disclosed