SCHEMBL7956853

SCHEMBL7956853

CCSc1n[nH]c(-c2c(Cl)cc(C(F)(F)F)c(N)c2Cl)c1C#N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 3/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 2/20 0.38
STAT6 P42226 1/20 0.38
HIF1A Q16665 1/20 0.38
LMNA P02545 1/20 0.33
GABRP O00591 2/20 0.33
GABRD O14764 2/20 0.33
GABRA1 P14867 2/20 0.33
GABRB1 P18505 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA5 P31644 2/20 0.33
GABRA3 P34903 2/20 0.33
GABRA2 P47869 2/20 0.33
GABRB2 P47870 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7957533 0.88 GABRP (0.41) KDM4EMEN1KMT2AALDH1A1MAPT
SCHEMBL7970339 0.83 RET (0.43) KDM4EALDH1A1POLBMAPTHPGD
SCHEMBL7969879 0.78 GLP1R (0.33) KDM4EMEN1KMT2AALDH1A1HPGD
SCHEMBL7973060 0.78 GRM5 (0.30) GRM5
SCHEMBL8302702 0.75 GABRP (0.32) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL7460779 0.74
SCHEMBL364961 0.73
SCHEMBL8507631 0.72
SCHEMBL8552313 0.71
SCHEMBL7970231 0.70 GABRP (0.42) MAPTGABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001007413-A1 1-ARYL-3-THIOALKYL PYRAZOLES, THE SYNTHESIS THEREOF AND THE USE THEREOF AS INSECTICIDES 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-02-01 WO claimed
WO-2001007413-A1 1-ARYL-3-THIOALKYL PYRAZOLES, THE SYNTHESIS THEREOF AND THE USE THEREOF AS INSECTICIDES 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-02-01 WO disclosed