SCHEMBL7957533

SCHEMBL7957533

CSc1n[nH]c(-c2c(Cl)cc(C(F)(F)F)c(N)c2Cl)c1C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 7/20 0.41
GABRD O14764 7/20 0.41
GABRA1 P14867 7/20 0.41
GABRB1 P18505 7/20 0.41
GABRG2 P18507 7/20 0.41
GABRB3 P28472 7/20 0.41
GABRA5 P31644 7/20 0.41
GABRA3 P34903 7/20 0.41
GABRA2 P47869 7/20 0.41
GABRB2 P47870 7/20 0.41
GABRA4 P48169 7/20 0.41
GABRE P78334 7/20 0.41
GABRA6 Q16445 7/20 0.41
GABRG1 Q8N1C3 7/20 0.41
GABRG3 Q99928 7/20 0.41
GABRQ Q9UN88 7/20 0.41
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7956853 0.88 KDM4E (0.38) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL8302702 0.82 GABRP (0.32) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL7966297 0.81 GABRP (0.51) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL7973060 0.81 GRM5 (0.30) GRM5
SCHEMBL7969879 0.81 GLP1R (0.33) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL7970339 0.80 RET (0.43) KDM4EALDH1A1L3MBTL1TDP1HPGD
SCHEMBL7970231 0.79 GABRP (0.42) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL7460779 0.76
SCHEMBL364961 0.76
SCHEMBL1644627 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001007413-A1 1-ARYL-3-THIOALKYL PYRAZOLES, THE SYNTHESIS THEREOF AND THE USE THEREOF AS INSECTICIDES 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-02-01 WO claimed
WO-2001007413-A1 1-ARYL-3-THIOALKYL PYRAZOLES, THE SYNTHESIS THEREOF AND THE USE THEREOF AS INSECTICIDES 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-02-01 WO disclosed