SCHEMBL7956978

SCHEMBL7956978

O=S1(=O)N=C(Cl)Nc2ccc(Br)cc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
THRB P10828 1/20 0.51
TSHR P16473 1/20 0.51
ABCC8 Q09428 1/20 0.51
KCNJ11 Q14654 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CA12 O43570 3/20 0.50
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
CA9 Q16790 3/20 0.50
CA4 P22748 2/20 0.50
CA7 P43166 2/20 0.50
CXCR2 P25025 5/20 0.39
TGM2 P21980 1/20 0.36
CES1 P23141 1/20 0.36
GABRA1 P14867 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30885705 0.86 ALDH1A1 (0.44) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL31734749 0.79 ABCC8 (0.51) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL7954653 0.79 CA12 (0.46) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
Water SCHEMBL7951041 0.78 CA12 (0.45) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL717082 0.78 CA1 (0.45) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL5627683 0.76 CA12 (0.44) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL7953074 0.74 CA12 (0.42) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL8493177 0.74 CA12 (0.42) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL22616509 0.74 CA12 (0.65) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL8488778 0.74 ALDH1A1 (0.43) ALDH1A1LMNACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1081633-C 1,2, 4-benzothiadiazine derivatives, method for preparing same and use thereof NOVO NORDISK AS (DK) 2002-03-27 CN disclosed
US-6242443-B1 1,2,4-benzothiadiazine derivatives, their preparation and use NOVO NORDISK AIS (DK) 2001-06-05 US disclosed
CN-1222910-A 1,2, 4-benzothiadiazine derivatives, method for preparing same and use thereof NOVO NORDISK AS (DK) 1999-07-14 CN disclosed