SCHEMBL7958461

SCHEMBL7958461

CC(C)n1cnc2c(=S)[nH]c(=O)[nH]c21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
PI4KA P42356 1/20 0.35
PI4K2B Q8TCG2 1/20 0.35
PI4K2A Q9BTU6 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
CDK1 P06493 3/20 0.34
CCNB1 P14635 2/20 0.34
CDK2 P24941 2/20 0.34
CCNE1 P24864 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10001264 0.83 MEN1 (0.45) ALDH1A1MEN1KMT2AADORA2AADORA2B
SCHEMBL15290224 0.78 ALDH1A1 (0.56) ALDH1A1MEN1KMT2AADORA2AADORA1
SCHEMBL5436105 0.77 ALDH1A1 (0.50) ALDH1A1MEN1KMT2AADORA2AADORA2B
SCHEMBL7416953 0.75 ALDH1A1 (0.47) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL17311159 0.75 ALDH1A1 (0.56) ALDH1A1TSHRCYP2C19HSD17B10
SCHEMBL7419700 0.74 ALDH1A1 (0.46) ALDH1A1KMT2ACDK2CCNE1
SCHEMBL1964476 0.73 ALDH1A1 (0.42) ALDH1A1
SCHEMBL9845196 0.72 ALDH1A1 (0.50) ALDH1A1KMT2AADORA2AADORA2BADORA1
SCHEMBL18510398 0.71 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AADORA2AADORA2B
SCHEMBL18510362 0.70 MEN1 (0.42) ALDH1A1MEN1KMT2AADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6268373-B1 ENZYME INHIBITORS EURO-CELTIQUE S.A. (LU) 2001-07-31 US disclosed