SCHEMBL7958501

SCHEMBL7958501

CN/C(N)=N\C1(C2CC2)CC(c2ccncc2)Oc2ccc(Br)cc21

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.35
BACE1 P56817 10/20 0.33
APP P05067 6/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16136607 0.67 AKR1B1 (0.35) AKR1B1BACE1APP
SCHEMBL1829170 0.67 BACE1 (0.43) AKR1B1BACE1APP
SCHEMBL16136524 0.62 AKR1B1 (0.38) AKR1B1BACE1
SCHEMBL12299265 0.61 AKR1B1 (0.37) AKR1B1BACE1
SCHEMBL12246365 0.61 AKR1B1 (0.46) AKR1B1
Hydrochloric Acid SCHEMBL1822716 0.60 AKR1B1 (0.45) AKR1B1
SCHEMBL1824431 0.59 AKR1B1 (0.42) AKR1B1
SCHEMBL1821217 0.58 AR (0.57)
SCHEMBL1822169 0.58 AKR1B1 (0.44) AKR1B1BACE1
SCHEMBL16230122 0.57 BACE1 (0.51) BACE1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed