SCHEMBL16136607

SCHEMBL16136607

CNC1=NC2(CC(c3ccncc3)Oc3ccc(Br)cc32)ON1C

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.35
BACE1 P56817 15/20 0.34
BACE2 Q9Y5Z0 1/20 0.34
CTSD P07339 2/20 0.33
APP P05067 5/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1829170 0.86 BACE1 (0.43) AKR1B1BACE1BACE2CTSDAPP
SCHEMBL1823750 0.76 BACE1 (0.53) AKR1B1BACE1BACE2CTSDAPP
SCHEMBL2374794 0.74 BACE1 (0.45) BACE1BACE2CTSDAPP
SCHEMBL7964852 0.72 BACE1 (0.31) AKR1B1BACE1
SCHEMBL1822145 0.71 BACE1 (0.41) AKR1B1BACE1BACE2CTSD
SCHEMBL1828177 0.69 BACE1 (0.44) BACE1CTSDAPP
SCHEMBL7969641 0.69 BACE1 (0.37) BACE1CTSDAPP
SCHEMBL1828027 0.68 ALOX12 (0.37) AKR1B1
SCHEMBL7948209 0.67 OPRM1 (0.39) AKR1B1
SCHEMBL7958501 0.67 AKR1B1 (0.35) AKR1B1BACE1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324032-B1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS INC (US) 2014-10-01 EP disclosed