SCHEMBL7959486

SCHEMBL7959486

O=C1C=C(c2ccccc2)C1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.52
RAB9A P51151 1/20 0.52
CFTR P13569 2/20 0.48
GOPC Q9HD26 2/20 0.48
ALDH1A1 P00352 3/20 0.46
LMNA P02545 2/20 0.46
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
CYP2A6 P11509 1/20 0.41
BACE1 P56817 1/20 0.41
HPGD P15428 1/20 0.40
AXL P30530 1/20 0.39
CTRC Q99895 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL731336 0.82 NPC1 (0.50) NPC1RAB9ACFTRGOPCALDH1A1
SCHEMBL679561 0.78 NPC1 (0.47) NPC1RAB9ACFTRGOPCALDH1A1
SCHEMBL27546185 0.74 ALDH1A1 (0.40) NPC1RAB9ACFTRGOPCALDH1A1
SCHEMBL29489303 0.73 FYN (0.42) RAB9AALDH1A1MAPTHPGDMAOB
SCHEMBL8902488 0.73 BACE1 (0.46) NPC1RAB9ACFTRGOPCALDH1A1
SCHEMBL8007243 0.72 NPC1 (0.93) NPC1RAB9AALDH1A1LMNAHPGD
SCHEMBL11180936 0.72 NPC1 (0.46) NPC1RAB9AALDH1A1LMNAHPGD
Biphenyl SCHEMBL15657385 0.71 ALDH1A1 (0.60) NPC1RAB9ACFTRGOPCALDH1A1
SCHEMBL28199530 0.70 CFTR (0.40) NPC1RAB9ACFTRGOPCALDH1A1
SCHEMBL602159 0.70 GSK3A (0.41) ALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114426510-A Synthesis method of fully-substituted beta-lactam 常州大学 2022-05-03 CN disclosed
WO-2012073038-A2 COMPOUNDS AND METHODS OF MAKING THE SAME UNIVERSITY OF SHEFFIELD (GB) 2012-06-07 WO disclosed
US-6291520-B1 INHIBIT THE ENZYME LIPOXYGENASE; TREATMENT OR ALLEVIATION OF INFLAMMATORY DISEASES, ALLERGIC CONDITIONS AND CARDIOVASCULAR DISEASES PFIZER 2001-09-18 US disclosed
EP-0559743-B1 NOVEL HYDROXAMIC ACID AND N-HYDROXYUREA DERIVATIVES AND THEIR USE PFIZER (US) 1995-03-08 EP disclosed
EP-0559743-A1 NOVEL HYDROXAMIC ACID AND N-HYDROXYUREA DERIVATIVES AND THEIR USE. PFIZER HOSPITAL PROD (US) 1993-09-15 EP disclosed
WO-1992009566-A1 NOVEL HYDROXAMIC ACID AND N-HYDROXYUREA DERIVATIVES AND THEIR USE PFIZER INC. (US) 1992-06-11 WO disclosed