SCHEMBL7960106

SCHEMBL7960106

CCOC(=O)N1CCC2(CC1)N=C(N)c1ncccc1N2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 8/20 0.67
NOS1 P29475 5/20 0.67
NOS3 P29474 2/20 0.67
HRH1 P35367 2/20 0.44
OPRD1 P41143 4/20 0.42
OPRK1 P41145 3/20 0.42
OPRM1 P35372 2/20 0.42
FAAH O00519 1/20 0.41
MGLL Q99685 1/20 0.41
SMO Q99835 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KCNH2 Q12809 3/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
MPI P34949 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7938165 0.84 NOS2 (0.70) NOS2NOS1NOS3OPRD1OPRK1
SCHEMBL7964756 0.83 NOS2 (0.59) NOS2NOS1NOS3HRH1OPRD1
Hydrochloric Acid SCHEMBL8379762 0.83 NOS2 (0.69) NOS2NOS1NOS3OPRD1OPRK1
SCHEMBL7938121 0.82 NOS2 (0.81) NOS2NOS1NOS3OPRD1OPRK1
Hydrochloric Acid SCHEMBL8381053 0.81 NOS2 (0.79) NOS2NOS1NOS3OPRD1OPRK1
SCHEMBL7940883 0.80 NOS2 (1.00) NOS2NOS1NOS3OPRD1KDM4E
SCHEMBL7940944 0.80 NOS2 (1.00) NOS2NOS1NOS3OPRD1OPRK1
SCHEMBL7940741 0.79 NOS2 (0.76) NOS2NOS1NOS3KDM4EALDH1A1
Hydrochloric Acid SCHEMBL8379951 0.79 NOS2 (0.98) NOS2NOS1NOS3OPRD1KDM4E
Hydrochloric Acid SCHEMBL8376957 0.79 NOS2 (0.98) NOS2NOS1NOS3OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303613-B1 AS NITRIC OXIDE SYNTHASE INHIBITOR USEFUL IN THERAPY OR PROPHYLAXIS OF INFLAMMATORY DISEASE AND PAIN ASTRAZENECA AB (SE) 2001-10-16 US disclosed