SCHEMBL7960345

SCHEMBL7960345

O=[N+]([O-])c1cc(Br)nc(N2CCNCC2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
HTR3E A5X5Y0 1/20 0.54
HTR3B O95264 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
SLC6A4 P31645 1/20 0.54
CYP2C19 P33261 1/20 0.54
THPO P40225 1/20 0.54
HTR3A P46098 1/20 0.54
HTR3D Q70Z44 1/20 0.54
HTR3C Q8WXA8 1/20 0.54
HTR1D P28221 1/20 0.51
HTR2C P28335 1/20 0.51
HTR6 P50406 1/20 0.51
ADRB1 P08588 1/20 0.49
SIRT6 Q8N6T7 1/20 0.49
LMNA P02545 1/20 0.46
PMP22 Q01453 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CASP1 P29466 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tert-Butyl Formate SCHEMBL27835007 0.86 ALDH1A1 (0.46) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL31401096 0.82 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2C19LMNA
SCHEMBL9318302 0.76 ALDH1A1 (0.64) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL6364738 0.75 ALDH1A1 (0.66) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL9069868 0.75 ALDH1A1 (0.59) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL31401459 0.74 KMT2A (0.35) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL31061212 0.73 ALDH1A1 (0.58) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL31263688 0.73 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP2C19LMNANPSR1
SCHEMBL21635259 0.73 GRIN2D (0.58)
SCHEMBL220662 0.73 CYP19A1 (0.50) ALDH1A1CYP1A2CYP3A4LMNAPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150230-A1 2,4'-BIPYRIDINYL COMPOUNDS AS PROTEIN KINASE D INHIBITORS USEFUL FOR THE TREATMENT OF IA HEART FAILURE AND CANCER NOVARTIS AG (CH) 2009-12-17 WO disclosed