SCHEMBL9318302

SCHEMBL9318302

O=[N+]([O-])c1cc(Br)c2nc(N3CCNCC3)ccc2c1

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.64
HTR3E A5X5Y0 2/20 0.64
HTR3B O95264 2/20 0.64
HTR3A P46098 2/20 0.64
HTR3D Q70Z44 2/20 0.64
HTR3C Q8WXA8 2/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
SLC6A4 P31645 1/20 0.64
CYP2C19 P33261 1/20 0.64
THPO P40225 1/20 0.64
LMNA P02545 1/20 0.55
PMP22 Q01453 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
ADRB1 P08588 1/20 0.46
SIRT6 Q8N6T7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
6-Nitroquipazine SCHEMBL401156 0.78 ALDH1A1 (1.00) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7960345 0.76 ALDH1A1 (0.54) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL9318631 0.75 ALDH1A1 (0.64) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL31060742 0.74 ALDH1A1 (0.90) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL3299921 0.73 HTR3A (0.58) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL6364738 0.72 ALDH1A1 (0.66) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4002581 0.72 ADRB1 (0.58) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL26650780 0.71 NQO2 (0.51) ALDH1A1CYP3A4
SCHEMBL31357879 0.71 NQO2 (0.55) ALDH1A1CYP3A4LMNANPSR1
6-Nitroquipazine SCHEMBL4266389 0.71 ALDH1A1 (1.00) ALDH1A1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5372813-A Measurement of serotonin uptake sites in a sample using a radio labeled substituted 6-nitroquipazine as a radioligand THE REGENTS, UNIVERSITY OF CALIFORNIA (US) 1994-12-13 US disclosed