SCHEMBL7962398

SCHEMBL7962398

O=C1NC(=S)S/C1=C\c1ccc(Cl)c(Cl)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAT1 P18440 7/20 1.00
IGF1R P08069 1/20 0.75
MYC P01106 3/20 0.70
MAX P61244 3/20 0.70
ADAMTS5 Q9UNA0 1/20 0.69
DNM1 Q05193 1/20 0.68
PTP4A3 O75365 1/20 0.63
CRHBP P24387 1/20 0.63
CRHR2 Q13324 1/20 0.63
MEN1 O00255 1/20 0.63
PIM1 P11309 1/20 0.63
RAB9A P51151 1/20 0.63
KMT2A Q03164 1/20 0.63
CISD1 Q9NZ45 2/20 0.61
CA2 P00918 1/20 0.60
EPHX1 P07099 1/20 0.60
PDE4B Q07343 1/20 0.60
PDE3A Q14432 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6781138 1.00 NAT1 (1.00) NAT1IGF1RMYCMAXADAMTS5
SCHEMBL12892058 1.00 NAT1 (1.00) NAT1IGF1RMYCMAXADAMTS5
SCHEMBL14381062 0.87 NAT1 (0.77) NAT1IGF1RMYCMAXDNM1
SCHEMBL6785380 0.86 IGF1R (1.00) NAT1IGF1RADAMTS5PIM1RAB9A
SCHEMBL6785383 0.86 IGF1R (1.00) NAT1IGF1RADAMTS5PIM1RAB9A
SCHEMBL1249067 0.83 NAT1 (1.00) NAT1MYCMAXDNM1CRHBP
SCHEMBL1249069 0.83 NAT1 (1.00) NAT1MYCMAXDNM1CRHBP
SCHEMBL20816059 0.83 NAT1 (1.00) NAT1MYCMAXDNM1CRHBP
SCHEMBL13499589 0.83 GSK3B (0.74) NAT1IGF1RMYCMAXADAMTS5
SCHEMBL7557495 0.82 ADAMTS5 (1.00) NAT1ADAMTS5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0343643-A2 Arylmethylenyl derivatives of thiazolidnones, imidazolidinones and oxazolidinones useful as antiallergy agents and antiinflamatory agents WARNER-LAMBERT COMPANY (US) 1989-11-29 EP claimed
US-8431376-B2 Bacterial replication systems and methods THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2013-04-30 US disclosed
US-8431376-B2 Bacterial replication systems and methods THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2013-04-30 US disclosed
US-20100028862-A1 BACTERIAL REPLICATION SYSTEMS AND METHODS Replidyne,Inc. (US) 2010-02-04 US disclosed
US-20100028862-A1 BACTERIAL REPLICATION SYSTEMS AND METHODS Replidyne,Inc. (US) 2010-02-04 US disclosed
WO-2006071255-A9 BACTERIAL REPLICATION SYSTEMS AND METHODS REPLIDYNE INC (US) 2007-02-15 WO disclosed
WO-2001077091-A2 NS5B HCV POLYMERASE INHIBITORS TULARIK INC. (US) 2001-10-18 WO disclosed
WO-2000018748-A1 RHODANINE DERIVATIVES FOR THE TREATMENT AND PREVENTION OF METABOLIC BONE DISORDERS ROCHE DIAGNOSTICS GMBH (DE) 2000-04-06 WO disclosed
EP-0915090-A1 Compounds useful as hypoglycemic agents and for treating Alzheimer's disease ELI LILLY AND COMPANY (US) 1999-05-12 EP disclosed
US-5716975-A NONTOXIC RHODANINE DERIVATIVES; ANTIDIABETIC AGENTS, CATHEPSIN D INHIBITORS, B-AMYLOID PROTEIN REDUCTION ELI LILLY AND COMPANY (US) 1998-02-10 US disclosed
US-5661168-A ADMINISTERING RHODANINE DERIVATIVES TO CONTROL DIABETES ELI LILLY AND COMPANY (US) 1997-08-26 US disclosed
US-5523314-A RHODANINE DERIVATIVES ELI LILLY AND COMPANY (US) 1996-06-04 US disclosed
US-5464856-A Arylmethylenyl derivatives of imidazolidinones useful as antiinflammatory agents WARNER-LAMBERT COMPANY (US) 1995-11-07 US disclosed
US-5306822-A Mono-, di- or tri-methoxyphenylmethylene-2-thioxo-4-oxazolidinone as antihistamines WARNER-LAMBERT COMPANY (US) 1994-04-26 US disclosed
EP-0587377-A2 Thiazolidinone derivatives as hypoglycemic agents and for treating Alzheimer's disease ELI LILLY AND COMPANY (US) 1994-03-16 EP disclosed
US-5208250-A Known and selected novel arylmethylenyl derivatives of thiazolidinones, imidazolidinones and oxazolidinones useful as antiallergy agents and anti-inflammatory agents WARNER-LAMBERT COMPANY (US) 1993-05-04 US disclosed
EP-0343643-A2 Arylmethylenyl derivatives of thiazolidnones, imidazolidinones and oxazolidinones useful as antiallergy agents and antiinflamatory agents WARNER-LAMBERT COMPANY (US) 1989-11-29 EP disclosed