SCHEMBL7962689

SCHEMBL7962689

COc1ccc2c(c1)N(CC(=O)C(C)(C)C)C(=O)C(NC(=O)OCc1ccccc1)CN2c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.40
BRD2 P25440 1/20 0.40
BRD3 Q15059 1/20 0.40
XIAP P98170 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ACHE P22303 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KCNQ2 O43526 1/20 0.38
TP53 P04637 1/20 0.37
CCKBR P32239 3/20 0.36
TSHR P16473 2/20 0.36
CYP3A4 P08684 1/20 0.36
PREP P48147 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6178982 0.90 ACE (0.41) ALDH1A1PREP
SCHEMBL6179084 0.85 CA1 (0.32) BRD4BRD2BRD3XIAPCA1
SCHEMBL7959523 0.81 TSHR (0.39) ALDH1A1TP53CCKBRTSHR
SCHEMBL6177308 0.80 PARP1 (0.40) ALDH1A1CCKBRPREP
SCHEMBL6177621 0.80 CCKBR (0.49) CCKBR
SCHEMBL6176498 0.79 CCKBR (0.44) CCKBR
SCHEMBL6179330 0.79 CCKBR (0.47) TP53CCKBRTSHR
SCHEMBL6176919 0.79 CCKBR (0.42) CCKBR
SCHEMBL17557005 0.78 CA1 (0.47) CA1CA2ACHEALDH1A1KCNQ2
SCHEMBL16059873 0.78 CA1 (0.47) CA1CA2ACHEALDH1A1KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed