SCHEMBL7959523

SCHEMBL7959523

COc1ccc2c(c1)N(CC(=O)C(C)(C)C)C(=O)C(N)CN2c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
KYAT1 Q16773 1/20 0.39
KYAT3 Q6YP21 1/20 0.39
AADAT Q8N5Z0 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 3/20 0.37
GRM2 Q14416 2/20 0.37
HTT P42858 1/20 0.37
CCKBR P32239 1/20 0.36
TP53 P04637 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
PDPK1 O15530 1/20 0.36
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
MAPT P10636 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6176017 0.87 CCKAR (0.39) AADATALDH1A1CCKBR
SCHEMBL1394353 0.86 ALDH1A1 (0.48) ALDH1A1CCKBR
SCHEMBL6176423 0.86 ALDH1A1 (0.48) ALDH1A1CCKBR
SCHEMBL7962381 0.83 KYAT1 (0.40) TSHRKYAT1KYAT3AADATALDH1A1
Oxalic Acid SCHEMBL6825172 0.83 ALDH1A1 (0.46) ALDH1A1CCKBR
Oxalic Acid SCHEMBL6825177 0.83 ALDH1A1 (0.46) ALDH1A1CCKBR
SCHEMBL7962689 0.81 BRD4 (0.40) TSHRALDH1A1CCKBRTP53
SCHEMBL6177621 0.78 CCKBR (0.49) CCKBR
SCHEMBL6178095 0.75 MAPT (0.42) CCKBRMAPT
SCHEMBL6179330 0.75 CCKBR (0.47) TSHRCCKBRTP53LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed